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MILLARD, CHRISTOPHER J, LUDEMAN, JUSTIN P, CANALS, MERITXELL, BRIDGFORD, JESSICA L, HINDS, MARK G, CLAYTON, DANIEL J, CHRISTOPOULOS, ARTHUR, PAYNE, RICHARD J and STONE, MARTIN J, 2014. Structural Basis of Receptor Sulfotyrosine Recognition by a CC Chemokine: The N-Terminal Region of CCR3 Bound to CCL11/Eotaxin-1 Structure. 22(11), 1571-1581 ABDUL-RIDHA, A, LANE, JR, MISTRY, SN, LOPEZ, L, SEXTON, PM, SCAMMELLS, PJ, CHRISTOPOULOS, A and CANALS, M, 2014. Mechanistic Insights into Allosteric Structure-Function Relationships at the M1 Muscarinic Acetylcholine Receptor Journal of Biological Chemistry. 289(48), 33701-33711 DROR, RON O, GREEN, HILLARY F, VALANT, CELINE, BORHANI, DAVID W, VALCOURT, JAMES R, PAN, ALBERT C, ARLOW, DANIEL H, CANALS, MERITXELL, LANE, J ROBERT, RAHMANI, RAPHAËL, BAELL, JONATHAN B, SEXTON, PATRICK M, CHRISTOPOULOS, ARTHUR and SHAW, DAVID E, 2013. Structural basis for modulation of a G-protein-coupled receptor by allosteric drugs. Nature. 503(7475), 295-299 SCHOLTEN, D J, ROUMEN, L, WIJTMANS, M, VERKADE-VREEKER, M C A, CUSTERS, H, LAI, M, DE HOOGE, D, CANALS, M, DE ESCH, I J P, SMIT, M J, DE GRAAF, C and LEURS, R, 2013. Identification of Overlapping but Differential Binding Sites for the High-Affinity CXCR3 Antagonists NBI-74330 and VUF11211 Mol Pharmacol. 85(1), 116-126 TAN, J H Y, LUDEMAN, J P, WEDDERBURN, J, CANALS, M, HALL, P, BUTLER, S J, TALESKI, D, CHRISTOPOULOS, A, HICKEY, M J, PAYNE, R J and STONE, M J, 2013. Tyrosine Sulfation of Chemokine Receptor CCR2 Enhances Interactions with Both Monomeric and Dimeric Forms of the Chemokine Monocyte Chemoattractant Protein-1 (MCP-1) The Journal of biological chemistry. 288(14), 10024-10034
JENSEN, DANE D, GODFREY, CODY B, NIKLAS, CHRISTIAN, CANALS, MERITXELL, KOCAN, MARTINA, POOLE, DANIEL P, MURPHY, JANE E, ALEMI, FARZAD, COTTRELL, GRAEME S, KORBMACHER, CHRISTOPH, LAMBERT, NEVIN A, BUNNETT, NIGEL W and CORVERA, CARLOS U, 2013. The bile acid receptor TGR5 does not interact with $beta$-arrestins or traffic to endosomes but transmits sustained signals from plasma membrane rafts. The Journal of biological chemistry. 288(32), 22942-22960
LANE, J ROBERT, ABDUL-RIDHA, ALAA and CANALS, MERITXELL, 2013. Regulation of G protein-coupled receptors by allosteric ligands ACS chemical neuroscience. 130212081603007 ZHAO, PEISHEN, CANALS, MERITXELL, MURPHY, JANE E, KLINGLER, DIANA, ERIKSSON, EMILY M, PELAYO, JUAN-CARLOS, HARDT, MARKUS, BUNNETT, NIGEL W and POOLE, DANIEL P, 2013. Agonist-biased Trafficking of Somatostatin Receptor 2A in Enteric Neurons. The Journal of biological chemistry. 288(36), 25689-25700
SCHOLTEN, D J, CANALS, M, WIJTMANS, M, DE MUNNIK, S, NGUYEN, P, VERZIJL, D, DE ESCH, I J P, VISCHER, H F, SMIT, M J and LEURS, R, 2012. Pharmacological characterization of a small-molecule agonist for the chemokine receptor CXCR3. British Journal of Pharmacology. 166(3), 898-911 ABDUL-RIDHA, A, LANE, J R, SEXTON, P M, CANALS, M and CHRISTOPOULOS, A, 2012. Allosteric Modulation of a Chemogenetically Modified G Protein-Coupled Receptor Mol Pharmacol. WIJTMANS, MAIKEL, SCHOLTEN, DANNY J, ROUMEN, LUC, CANALS, MERITXELL, CUSTERS, HANS, GLAS, MARJOLEIN, VREEKER, MARLIES C A, DE KANTER, FRANS J J, DE GRAAF, CHRIS, SMIT, MARTINE J, DE ESCH, IWAN J P and LEURS, ROB, 2012. Chemical Subtleties in Small-Molecule Modulation of Peptide Receptor Function: The Case of CXCR3 Biaryl-Type Ligands Journal of Medicinal Chemistry. 121114090531003 CANALS, MERITXELL, SCHOLTEN, DANNY J, DE MUNNIK, SABRINA, HAN, MITCHELL K L, SMIT, MARTINE J and LEURS, ROB, 2012. Ubiquitination of CXCR7 controls receptor trafficking. PLoS ONE. 7(3), e34192 CANALS, MERITXELL, LANE, J ROBERT, WEN, ADRIEL, SCAMMELLS, PETER J, SEXTON, PATRICK M and CHRISTOPOULOS, ARTHUR, 2012. A Monod-Wyman-Changeux Mechanism Can Explain G Protein-coupled Receptor (GPCR) Allosteric Modulation. The Journal of biological chemistry. 287(1), 650-659
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